FAIRMol

OSA_Lib_77

Pose ID 1007 Compound 308 Pose 1007

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.465 kcal/mol/HA) ✓ Good fit quality (FQ -4.65) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (27.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-15.815
kcal/mol
LE
-0.465
kcal/mol/HA
Fit Quality
-4.65
FQ (Leeson)
HAC
34
heavy atoms
MW
465
Da
LogP
1.20
cLogP
Strain ΔE
27.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 27.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 1 Clashes 17 Severe clashes 2
Final rank60.38065659113832Score-15.815
Inter norm-0.565567Intra norm0.100421
Top1000noExcludedyes
Contacts18H-bonds5
Artifact reasonexcluded; geometry warning; 16 clashes; 2 protein clashes
ResiduesA:ALA10;A:ASN65;A:ASP22;A:GLU31;A:GLY21;A:ILE8;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TRP25;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap15Native recall0.71
Jaccard0.62RMSD-
H-bond strict2Strict recall0.40
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
980 4.2667967127332425 -0.647076 -18.8906 1 17 0 0.00 0.00 - no Open
964 4.4375082130399335 -0.666507 -20.7389 1 17 0 0.00 0.00 - no Open
963 4.8283277279898265 -0.818882 -26.4773 0 22 0 0.00 0.00 - no Open
976 4.861076246789533 -0.717485 -23.0849 3 19 0 0.00 0.00 - no Open
1020 5.608822815282937 -0.559562 -18.2789 2 17 13 0.62 0.00 - no Open
975 5.658661119979025 -0.72701 -19.9178 3 16 0 0.00 0.00 - no Open
972 5.872917234042555 -0.66726 -10.5276 2 16 0 0.00 0.00 - no Open
1017 5.943411109675365 -0.558633 -16.3741 1 15 13 0.62 0.00 - no Open
1013 6.307109152626905 -0.591976 -22.2418 4 17 13 0.62 0.40 - no Open
998 6.617839771151886 -0.692384 -24.2271 4 22 18 0.86 0.60 - no Open
1005 7.263428324635448 -0.598723 -20.9956 0 17 16 0.76 0.00 - no Open
1001 8.518952245362764 -0.512154 -10.4528 2 19 15 0.71 0.00 - no Open
965 54.268108346420284 -0.680293 -21.6517 1 15 0 0.00 0.00 - no Open
969 54.730108154157584 -0.83792 -26.6193 2 19 0 0.00 0.00 - no Open
966 54.90998971603653 -0.681929 -20.9942 2 18 0 0.00 0.00 - no Open
974 55.25225600517029 -0.712966 -21.7259 2 17 0 0.00 0.00 - no Open
957 55.33920843725555 -0.601959 -15.7833 1 17 0 0.00 0.00 - no Open
961 55.34723382073465 -0.695261 -21.8508 1 19 0 0.00 0.00 - no Open
1018 55.577770402172845 -0.615158 -14.106 2 15 12 0.57 0.40 - no Open
970 56.763655045820364 -0.680825 -21.5861 1 17 0 0.00 0.00 - no Open
1015 55.7401178962693 -0.644859 -23.9105 4 18 18 0.86 0.40 - yes Open
979 56.22693303779636 -0.793334 -24.9168 1 22 0 0.00 0.00 - yes Open
959 56.22887233234621 -0.657743 -14.235 6 18 0 0.00 0.00 - yes Open
971 56.25495307434291 -0.857331 -26.9352 1 21 0 0.00 0.00 - yes Open
1014 56.3140252935371 -0.690966 -20.8452 2 22 18 0.86 0.20 - yes Open
999 56.37188078468921 -0.631895 -19.5435 1 19 16 0.76 0.00 - yes Open
973 56.56725214004422 -0.623201 -24.1552 1 15 0 0.00 0.00 - yes Open
968 56.7475004943868 -0.581465 -19.5245 6 18 0 0.00 0.00 - yes Open
967 56.759649217372015 -0.676006 -18.7339 3 20 0 0.00 0.00 - yes Open
978 57.32083151732589 -0.712682 -25.1394 4 20 0 0.00 0.00 - yes Open
997 57.3249242113801 -0.604676 -18.5954 4 17 14 0.67 0.40 - yes Open
1009 57.394715812575434 -0.52356 -11.3693 2 16 12 0.57 0.20 - yes Open
1002 57.4808605706708 -0.617815 -16.9265 5 18 16 0.76 0.20 - yes Open
1000 57.625401861715766 -0.674365 -18.6906 4 18 17 0.81 0.60 - yes Open
1019 57.800249436248784 -0.723992 -26.6835 1 24 20 0.95 0.20 - yes Open
958 57.93847770081955 -0.710876 -22.6368 2 17 0 0.00 0.00 - yes Open
1003 58.20546004129062 -0.675781 -24.2705 2 24 20 0.95 0.20 - yes Open
1006 58.38086441393017 -0.693607 -24.2081 5 21 18 0.86 0.60 - yes Open
977 58.49646276358023 -0.732312 -24.1209 2 15 0 0.00 0.00 - yes Open
1012 58.925483999481 -0.743273 -20.6742 3 19 17 0.81 0.00 - yes Open
1016 59.78910891302541 -0.540698 -18.6917 4 19 19 0.90 0.20 - yes Open
1011 59.83248892398216 -0.718821 -24.3108 3 20 17 0.81 0.00 - yes Open
1004 59.87167927601356 -0.603058 -21.4062 2 20 18 0.86 0.00 - yes Open
962 59.872548927288754 -0.784707 -24.1046 2 16 0 0.00 0.00 - yes Open
1008 60.23140483524128 -0.615151 -10.199 0 19 17 0.81 0.00 - yes Open
1007 60.38065659113832 -0.565567 -15.815 5 18 15 0.71 0.40 - yes Current
1010 60.75011301860987 -0.623404 -16.21 1 20 18 0.86 0.00 - yes Open
960 62.283215330865104 -0.611563 -6.28831 4 22 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -15.815kcal/mol
Ligand efficiency (LE) -0.4651kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.654
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 464.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.20
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 27.24kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 109.80kcal/mol
Minimised FF energy 82.56kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.