FAIRMol

Z19456272

ID 100

DB SELECTIONThis detail page is pinned to the current database context.
2D structure

SMILES: O=S(=O)(c1cccc(CSc2nnc(-c3ccc4c(c3)OCO4)o2)c1)N1CCOCC1

Formula: C20H19N3O6S2 | MW: 461.52100000000036

LogP: 2.778500000000001 | TPSA: 103.99000000000001

HBA/HBD: 9/- | RotB: 6

InChIKey: ADNYXMUCYMCKQX-UHFFFAOYSA-N

Recognized patterns

Click a named motif to highlight it in the 2D depiction or launch reverse search.
Highlighted: 1 pattern Pyridine Clear highlight

Properties

NameValueUnit
DOCK_BASE_INTER_RANK-0.848599-
DOCK_BASE_INTER_RANK-0.848148-
DOCK_BASE_INTER_RANK-0.940039-
DOCK_BASE_INTER_RANK-0.856427-
DOCK_BASE_INTER_RANK-0.811185-
DOCK_BASE_INTER_RANK-0.989791-
DOCK_BASE_INTER_RANK-0.874039-
DOCK_BASE_INTER_RANK-0.908661-
DOCK_BASE_INTER_RANK-0.949521-
DOCK_BASE_INTER_RANK-0.950541-
DOCK_BASE_INTER_RANK-0.882026-
DOCK_BASE_INTER_RANK-0.897555-
DOCK_BASE_INTER_RANK-1.008350-
DOCK_BASE_INTER_RANK-0.767307-
DOCK_BASE_INTER_RANK-0.829303-
DOCK_BASE_INTER_RANK-0.773608-
DOCK_BASE_INTER_RANK-0.732121-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_BOND_LENGTH_OUTLIERS0.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CLASH_COUNT8.000000-
DOCK_CLASH_COUNT10.000000-
DOCK_CLASH_COUNT8.000000-
DOCK_CLASH_COUNT10.000000-
DOCK_CLASH_COUNT8.000000-
DOCK_CLASH_COUNT8.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CLASH_COUNT8.000000-
DOCK_CLASH_COUNT8.000000-
DOCK_CLASH_COUNT10.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CLASH_COUNT10.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CLASH_COUNT9.000000-
DOCK_CONTACT_COUNT16.000000-
DOCK_CONTACT_COUNT19.000000-
DOCK_CONTACT_COUNT14.000000-
DOCK_CONTACT_COUNT13.000000-
DOCK_CONTACT_COUNT14.000000-
DOCK_CONTACT_COUNT13.000000-
DOCK_CONTACT_COUNT17.000000-
DOCK_CONTACT_COUNT15.000000-
DOCK_CONTACT_COUNT16.000000-
DOCK_CONTACT_COUNT15.000000-
DOCK_CONTACT_COUNT16.000000-
DOCK_CONTACT_COUNT10.000000-
DOCK_CONTACT_COUNT19.000000-
DOCK_CONTACT_COUNT15.000000-
DOCK_CONTACT_COUNT14.000000-
DOCK_CONTACT_COUNT12.000000-
DOCK_CONTACT_COUNT16.000000-
DOCK_EXPERIMENTT01-
DOCK_EXPERIMENTT02-
DOCK_EXPERIMENTT03-
DOCK_EXPERIMENTT03-
DOCK_EXPERIMENTT04-
DOCK_EXPERIMENTT05-
DOCK_EXPERIMENTT09-
DOCK_EXPERIMENTT10-
DOCK_EXPERIMENTT10-
DOCK_EXPERIMENTT10-
DOCK_EXPERIMENTT12-
DOCK_EXPERIMENTT12-
DOCK_EXPERIMENTT13-
DOCK_EXPERIMENTT15-
DOCK_EXPERIMENTT16-
DOCK_EXPERIMENTT16-
DOCK_EXPERIMENTT17-
DOCK_EXPERIMENT_ID1-
DOCK_EXPERIMENT_ID2-
DOCK_EXPERIMENT_ID3-
DOCK_EXPERIMENT_ID3-
DOCK_EXPERIMENT_ID4-
DOCK_EXPERIMENT_ID5-
DOCK_EXPERIMENT_ID9-
DOCK_EXPERIMENT_ID10-
DOCK_EXPERIMENT_ID10-
DOCK_EXPERIMENT_ID10-
DOCK_EXPERIMENT_ID12-
DOCK_EXPERIMENT_ID12-
DOCK_EXPERIMENT_ID13-
DOCK_EXPERIMENT_ID15-
DOCK_EXPERIMENT_ID16-
DOCK_EXPERIMENT_ID16-
DOCK_EXPERIMENT_ID17-
DOCK_FINAL_RANK0.954473-
DOCK_FINAL_RANK1.374105-
DOCK_FINAL_RANK1.805802-
DOCK_FINAL_RANK2.099488-
DOCK_FINAL_RANK0.270979-
DOCK_FINAL_RANK4.484717-
DOCK_FINAL_RANK2.283221-
DOCK_FINAL_RANK2.831215-
DOCK_FINAL_RANK2.986601-
DOCK_FINAL_RANK3.572589-
DOCK_FINAL_RANK2.859116-
DOCK_FINAL_RANK3.588860-
DOCK_FINAL_RANK3.435617-
DOCK_FINAL_RANK1.800777-
DOCK_FINAL_RANK2.018218-
DOCK_FINAL_RANK2.939096-
DOCK_FINAL_RANK1.219650-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOMETRY_ALERTwarning-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_GEOM_OK0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_HARD_GEOMETRY_FAIL0-
DOCK_IFP::A:ALA101-
DOCK_IFP::A:ALA101-
DOCK_IFP::A:ALA1111-
DOCK_IFP::A:ALA151-
DOCK_IFP::A:ALA151-
DOCK_IFP::A:ALA151-
DOCK_IFP::A:ALA2091-
DOCK_IFP::A:ALA2091-
DOCK_IFP::A:ALA2841-
DOCK_IFP::A:ALA671-
DOCK_IFP::A:ALA901-
DOCK_IFP::A:ALA901-
DOCK_IFP::A:ALA901-
DOCK_IFP::A:ARG1161-
DOCK_IFP::A:ARG1161-
DOCK_IFP::A:ARG1161-
DOCK_IFP::A:ARG1401-
DOCK_IFP::A:ARG1401-
DOCK_IFP::A:ARG1401-
DOCK_IFP::A:ARG1401-
DOCK_IFP::A:ARG1401-
DOCK_IFP::A:ARG1441-
DOCK_IFP::A:ARG1441-
DOCK_IFP::A:ARG1441-
DOCK_IFP::A:ARG1441-
DOCK_IFP::A:ARG1441-
DOCK_IFP::A:ARG1541-
DOCK_IFP::A:ARG171-
DOCK_IFP::A:ARG171-
DOCK_IFP::A:ARG2281-
DOCK_IFP::A:ARG2771-
DOCK_IFP::A:ARG2871-
DOCK_IFP::A:ARG291-
DOCK_IFP::A:ARG481-
DOCK_IFP::A:ARG971-
DOCK_IFP::A:ARG971-
DOCK_IFP::A:ASN1061-
DOCK_IFP::A:ASN1061-
DOCK_IFP::A:ASN1061-
DOCK_IFP::A:ASN1061-
DOCK_IFP::A:ASN1121-
DOCK_IFP::A:ASN911-
DOCK_IFP::A:ASN911-
DOCK_IFP::A:ASP131-
DOCK_IFP::A:ASP131-
DOCK_IFP::A:ASP131-
DOCK_IFP::A:ASP221-
DOCK_IFP::A:ASP2321-
DOCK_IFP::A:ASP3321-
DOCK_IFP::A:ASP521-
DOCK_IFP::A:ASP521-
DOCK_IFP::A:CYS721-
DOCK_IFP::A:CYS721-
DOCK_IFP::A:CYS721-
DOCK_IFP::A:GLN1041-
DOCK_IFP::A:GLU1381-
DOCK_IFP::A:GLU2741-
DOCK_IFP::A:GLU311-
DOCK_IFP::A:GLU311-
DOCK_IFP::A:GLY1961-
DOCK_IFP::A:GLY1971-
DOCK_IFP::A:GLY211-
DOCK_IFP::A:GLY2141-
DOCK_IFP::A:GLY2141-
DOCK_IFP::A:GLY2151-
DOCK_IFP::A:GLY2151-
DOCK_IFP::A:GLY2251-
DOCK_IFP::A:GLY2351-
DOCK_IFP::A:GLY2361-
DOCK_IFP::A:GLY2371-
DOCK_IFP::A:GLY2761-
DOCK_IFP::A:GLY2861-
DOCK_IFP::A:GLY731-
DOCK_IFP::A:GLY731-
DOCK_IFP::A:GLY731-
DOCK_IFP::A:HIS1051-
DOCK_IFP::A:HIS1051-
DOCK_IFP::A:HIS1051-
DOCK_IFP::A:HIS1051-
DOCK_IFP::A:HIS1051-
DOCK_IFP::A:HIS141-
DOCK_IFP::A:HIS141-
DOCK_IFP::A:HIS141-
DOCK_IFP::A:HIS1411-
DOCK_IFP::A:HIS1411-
DOCK_IFP::A:HIS1411-
DOCK_IFP::A:HIS1411-
DOCK_IFP::A:HIS1411-
DOCK_IFP::A:HIS1971-
DOCK_IFP::A:HIS2411-
DOCK_IFP::A:HIS2411-
DOCK_IFP::A:ILE1991-
DOCK_IFP::A:ILE2851-
DOCK_IFP::A:ILE451-
DOCK_IFP::A:ILE451-
DOCK_IFP::A:ILE611-
DOCK_IFP::A:ILE611-
DOCK_IFP::A:ILE81-
DOCK_IFP::A:LEU1011-
DOCK_IFP::A:LEU1011-
DOCK_IFP::A:LEU1361-
DOCK_IFP::A:LEU1361-
DOCK_IFP::A:LEU1881-
DOCK_IFP::A:LEU1881-
DOCK_IFP::A:LEU2261-
DOCK_IFP::A:LEU2261-
DOCK_IFP::A:LEU2271-
DOCK_IFP::A:LEU2291-
DOCK_IFP::A:LEU2291-
DOCK_IFP::A:LEU231-
DOCK_IFP::A:LEU231-
DOCK_IFP::A:LEU281-
DOCK_IFP::A:LEU281-
DOCK_IFP::A:LEU3321-
DOCK_IFP::A:LEU3341-
DOCK_IFP::A:LEU681-
DOCK_IFP::A:LEU941-
DOCK_IFP::A:LEU941-
DOCK_IFP::A:LYS2111-
DOCK_IFP::A:LYS2111-
DOCK_IFP::A:LYS571-
DOCK_IFP::A:LYS571-
DOCK_IFP::A:LYS691-
DOCK_IFP::A:LYS891-
DOCK_IFP::A:LYS891-
DOCK_IFP::A:LYS931-
DOCK_IFP::A:LYS931-
DOCK_IFP::A:LYS951-
DOCK_IFP::A:LYS951-
DOCK_IFP::A:MET1011-
DOCK_IFP::A:MET2331-
DOCK_IFP::A:MET3331-
DOCK_IFP::A:MET531-
DOCK_IFP::A:MET531-
DOCK_IFP::A:NAP2011-
DOCK_IFP::A:NAP2011-
DOCK_IFP::A:NDP3011-
DOCK_IFP::A:NDP3011-
DOCK_IFP::A:NDP3021-
DOCK_IFP::A:NDP3021-
DOCK_IFP::A:PHE1131-
DOCK_IFP::A:PHE1131-
DOCK_IFP::A:PHE1701-
DOCK_IFP::A:PHE1981-
DOCK_IFP::A:PHE2301-
DOCK_IFP::A:PHE321-
DOCK_IFP::A:PHE321-
DOCK_IFP::A:PHE351-
DOCK_IFP::A:PHE351-
DOCK_IFP::A:PHE561-
DOCK_IFP::A:PHE561-
DOCK_IFP::A:PHE911-
DOCK_IFP::A:PHE911-
DOCK_IFP::A:PRO1131-
DOCK_IFP::A:PRO1871-
DOCK_IFP::A:PRO2121-
DOCK_IFP::A:PRO2121-
DOCK_IFP::A:PRO2131-
DOCK_IFP::A:PRO2131-
DOCK_IFP::A:PRO271-
DOCK_IFP::A:PRO271-
DOCK_IFP::A:PRO621-
DOCK_IFP::A:PRO881-
DOCK_IFP::A:SER1111-
DOCK_IFP::A:SER1111-
DOCK_IFP::A:SER1121-
DOCK_IFP::A:SER2001-
DOCK_IFP::A:SER2001-
DOCK_IFP::A:SER3641-
DOCK_IFP::A:SER601-
DOCK_IFP::A:SER861-
DOCK_IFP::A:THR1171-
DOCK_IFP::A:THR1371-
DOCK_IFP::A:THR571-
DOCK_IFP::A:THR741-
DOCK_IFP::A:THR741-
DOCK_IFP::A:THR741-
DOCK_IFP::A:THR831-
DOCK_IFP::A:TRP251-
DOCK_IFP::A:TRP251-
DOCK_IFP::A:TRP471-
DOCK_IFP::A:TRP921-
DOCK_IFP::A:TRP921-
DOCK_IFP::A:TYR1141-
DOCK_IFP::A:TYR1221-
DOCK_IFP::A:TYR1911-
DOCK_IFP::A:TYR1941-
DOCK_IFP::A:TYR1941-
DOCK_IFP::A:TYR2101-
DOCK_IFP::A:TYR3311-
DOCK_IFP::A:TYR341-
DOCK_IFP::A:TYR3891-
DOCK_IFP::A:TYR491-
DOCK_IFP::A:TYR491-
DOCK_IFP::A:TYR491-
DOCK_IFP::A:TYR971-
DOCK_IFP::A:VAL1161-
DOCK_IFP::A:VAL1161-
DOCK_IFP::A:VAL1561-
DOCK_IFP::A:VAL2301-
DOCK_IFP::A:VAL2301-
DOCK_IFP::A:VAL491-
DOCK_IFP::A:VAL871-
DOCK_IFP::A:VAL881-
DOCK_IFP::A:VAL881-
DOCK_IFP::A:VAL91-
DOCK_IFP::A:VAL91-
DOCK_IFP::B:ALA2091-
DOCK_IFP::B:ALA321-
DOCK_IFP::B:ALA901-
DOCK_IFP::B:ARG1161-
DOCK_IFP::B:ARG461-
DOCK_IFP::B:ARG461-
DOCK_IFP::B:ARG481-
DOCK_IFP::B:ARG741-
DOCK_IFP::B:ASN2081-
DOCK_IFP::B:ASN2451-
DOCK_IFP::B:ASP131-
DOCK_IFP::B:ASP521-
DOCK_IFP::B:CYS721-
DOCK_IFP::B:GLY2141-
DOCK_IFP::B:GLY2151-
DOCK_IFP::B:GLY2461-
DOCK_IFP::B:GLY731-
DOCK_IFP::B:GLY731-
DOCK_IFP::B:GLY771-
DOCK_IFP::B:HIS141-
DOCK_IFP::B:HIS141-
DOCK_IFP::B:ILE151-
DOCK_IFP::B:ILE151-
DOCK_IFP::B:ILE451-
DOCK_IFP::B:ILE761-
DOCK_IFP::B:LEU731-
DOCK_IFP::B:LYS2111-
DOCK_IFP::B:LYS891-
DOCK_IFP::B:MET531-
DOCK_IFP::B:MET701-
DOCK_IFP::B:PHE561-
DOCK_IFP::B:PRO2121-
DOCK_IFP::B:PRO2131-
DOCK_IFP::B:PRO881-
DOCK_IFP::B:SER441-
DOCK_IFP::B:SER741-
DOCK_IFP::B:SER861-
DOCK_IFP::B:TRP471-
DOCK_IFP::B:TYR1621-
DOCK_IFP::B:TYR491-
DOCK_IFP::B:VAL1561-
DOCK_IFP::B:VAL301-
DOCK_IFP::B:VAL311-
DOCK_IFP::B:VAL491-
DOCK_IFP::B:VAL871-
DOCK_IFP::B:VAL881-
DOCK_IFP::D:ARG2871-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_IMPORT_SCOPEbest_by_name-
DOCK_MAX_CLASH_OVERLAP0.641633-
DOCK_MAX_CLASH_OVERLAP0.641644-
DOCK_MAX_CLASH_OVERLAP0.641868-
DOCK_MAX_CLASH_OVERLAP0.641575-
DOCK_MAX_CLASH_OVERLAP0.641618-
DOCK_MAX_CLASH_OVERLAP0.641621-
DOCK_MAX_CLASH_OVERLAP0.641841-
DOCK_MAX_CLASH_OVERLAP0.641644-
DOCK_MAX_CLASH_OVERLAP0.641874-
DOCK_MAX_CLASH_OVERLAP0.641873-
DOCK_MAX_CLASH_OVERLAP0.641670-
DOCK_MAX_CLASH_OVERLAP0.641776-
DOCK_MAX_CLASH_OVERLAP0.641586-
DOCK_MAX_CLASH_OVERLAP0.641801-
DOCK_MAX_CLASH_OVERLAP0.641770-
DOCK_MAX_CLASH_OVERLAP0.641665-
DOCK_MAX_CLASH_OVERLAP0.641806-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT2-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT3-
DOCK_POSE_COUNT2-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT1-
DOCK_POSE_COUNT2-
DOCK_POSE_COUNT1-
DOCK_PRE_RANK0.932559-
DOCK_PRE_RANK1.349847-
DOCK_PRE_RANK1.775841-
DOCK_PRE_RANK2.075136-
DOCK_PRE_RANK0.247468-
DOCK_PRE_RANK4.464076-
DOCK_PRE_RANK2.256767-
DOCK_PRE_RANK2.805086-
DOCK_PRE_RANK2.959696-
DOCK_PRE_RANK3.542427-
DOCK_PRE_RANK2.833941-
DOCK_PRE_RANK3.552615-
DOCK_PRE_RANK3.413265-
DOCK_PRE_RANK1.770431-
DOCK_PRE_RANK1.988212-
DOCK_PRE_RANK2.909816-
DOCK_PRE_RANK1.192135-
DOCK_PRIMARY_POSE_ID513-
DOCK_PRIMARY_POSE_ID1184-
DOCK_PRIMARY_POSE_ID1840-
DOCK_PRIMARY_POSE_ID2491-
DOCK_PRIMARY_POSE_ID3135-
DOCK_PRIMARY_POSE_ID5523-
DOCK_PRIMARY_POSE_ID6187-
DOCK_PRIMARY_POSE_ID7541-
DOCK_PRIMARY_POSE_ID8580-
DOCK_PRIMARY_POSE_ID9600-
DOCK_PRIMARY_POSE_ID10690-
DOCK_PRIMARY_POSE_ID10982-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_RANKING_MODEinter_strain_penalized-
DOCK_REPORT_IDselection_import_t01-
DOCK_REPORT_IDselection_import_t02-
DOCK_REPORT_IDselection_import_t03-
DOCK_REPORT_IDselection_import_t03-
DOCK_REPORT_IDselection_import_t04-
DOCK_REPORT_IDselection_import_t05-
DOCK_REPORT_IDselection_import_t09-
DOCK_REPORT_IDselection_import_t10-
DOCK_REPORT_IDselection_import_t10-
DOCK_REPORT_IDselection_import_t10-
DOCK_REPORT_IDselection_import_t12-
DOCK_REPORT_IDselection_import_t12-
DOCK_REPORT_IDselection_import_t13-
DOCK_REPORT_IDselection_import_t15-
DOCK_REPORT_IDselection_import_t16-
DOCK_REPORT_IDselection_import_t16-
DOCK_REPORT_IDselection_import_t17-
DOCK_RESIDUE_CONTACTSA:ALA10;A:ASP22;A:GLU31;A:GLY21;A:ILE61;A:LEU23;A:LEU28;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:TRP25;A:VAL116;A:VAL9-
DOCK_RESIDUE_CONTACTSA:ALA10;A:ARG29;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:THR137;A:THR57;A:TRP25;A:TYR122;A:TYR34;A:VAL116;A:VAL9-
DOCK_RESIDUE_CONTACTSA:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:SER86;A:THR83;A:VAL156;A:VAL87-
DOCK_RESIDUE_CONTACTSA:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO88;A:TRP47;A:VAL49-
DOCK_RESIDUE_CONTACTSA:ARG17;A:ASP232;A:GLY225;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:MET233;A:NDP302;A:PHE113;A:SER111;A:TYR191;A:TYR194;A:VAL230-
DOCK_RESIDUE_CONTACTSA:ARG17;A:HIS241;A:LEU188;A:LEU226;A:LEU229;A:NDP302;A:PHE113;A:SER111;A:SER112;A:TYR114;A:TYR194;A:VAL230;D:ARG287-
DOCK_RESIDUE_CONTACTSA:NDP301;B:ALA32;B:ARG48;B:ASP52;B:ILE45;B:MET53;B:PHE56;B:PRO88;B:SER44;B:SER86;B:TRP47;B:TYR162;B:VAL156;B:VAL30;B:VAL31;B:VAL49;B:VAL87-
DOCK_RESIDUE_CONTACTSA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLU138;A:GLY73;A:HIS105;A:HIS14;A:HIS141;A:LEU136;A:THR74;A:TYR49-
DOCK_RESIDUE_CONTACTSA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLN104;A:GLY73;A:HIS105;A:HIS14;A:HIS141;A:LEU101;A:LEU136;A:THR74;A:TYR49-
DOCK_RESIDUE_CONTACTSA:ALA15;A:ARG116;A:ARG140;A:ARG144;A:ASN106;A:ASP13;A:CYS72;A:GLY73;A:HIS105;A:HIS14;A:HIS141;A:LEU101;A:THR117;A:THR74;A:TYR49-
DOCK_RESIDUE_CONTACTSA:ARG140;A:ARG144;A:ASN106;A:HIS105;A:HIS141;A:MET101;B:ARG46;B:ASP13;B:CYS72;B:GLY73;B:GLY77;B:HIS14;B:ILE15;B:ILE76;B:SER74;B:TYR49-
DOCK_RESIDUE_CONTACTSA:ARG140;A:ARG144;A:HIS105;A:HIS141;A:TYR97;B:ARG116;B:ARG46;B:GLY73;B:HIS14;B:ILE15-
DOCK_RESIDUE_CONTACTSA:ALA111;A:ALA67;A:ALA90;A:ARG154;A:ARG277;A:ASN112;A:ASP332;A:GLU274;A:GLY235;A:GLY236;A:GLY237;A:GLY276;A:HIS197;A:LYS69;A:PHE170;A:PRO113;A:SER200;A:TYR331;A:TYR389-
DOCK_RESIDUE_CONTACTSB:ALA209;B:ALA90;B:ARG74;B:ASN208;B:ASN245;B:GLY214;B:GLY215;B:GLY246;B:LEU73;B:LYS211;B:LYS89;B:MET70;B:PRO212;B:PRO213;B:VAL88-
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DOCK_RESIDUE_CONTACTSA:ALA209;A:ALA90;A:ASN91;A:GLY214;A:GLY215;A:LYS211;A:LYS89;A:LYS93;A:PRO212;A:PRO213;A:TRP92;A:VAL88-
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DOCK_SOURCE_LOGP2.778500-
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DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_LOGP2.778500-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_MW461.521000-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEKB_Leish_4-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEKB_Leish_4-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEKB_Leish_4-
DOCK_SOURCE_NAMEKB_chagas_7-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEKB_Leish_4-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEKB_Leish_4-
DOCK_SOURCE_NAMEKB_chagas_7-
DOCK_SOURCE_NAMEZ19456272-
DOCK_SOURCE_NAMEKB_chagas_7-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_RINGS5.000000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_SOURCE_TPSA103.990000-
DOCK_STRAIN_DELTA17.585045-
DOCK_STRAIN_DELTA19.457398-
DOCK_STRAIN_DELTA23.523217-
DOCK_STRAIN_DELTA19.529760-
DOCK_STRAIN_DELTA18.876043-
DOCK_STRAIN_DELTA16.504623-
DOCK_STRAIN_DELTA21.095421-
DOCK_STRAIN_DELTA20.859082-
DOCK_STRAIN_DELTA21.419029-
DOCK_STRAIN_DELTA23.656346-
DOCK_STRAIN_DELTA20.153664-
DOCK_STRAIN_DELTA27.438732-
DOCK_STRAIN_DELTA17.945852-
DOCK_STRAIN_DELTA23.777499-
DOCK_STRAIN_DELTA23.552651-
DOCK_STRAIN_DELTA23.068122-
DOCK_STRAIN_DELTA21.852522-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_STRAIN_OK1-
DOCK_TARGETT01-
DOCK_TARGETT02-
DOCK_TARGETT03-
DOCK_TARGETT03-
DOCK_TARGETT04-
DOCK_TARGETT05-
DOCK_TARGETT09-
DOCK_TARGETT10-
DOCK_TARGETT10-
DOCK_TARGETT10-
DOCK_TARGETT12-
DOCK_TARGETT12-
DOCK_TARGETT13-
DOCK_TARGETT15-
DOCK_TARGETT16-
DOCK_TARGETT16-
DOCK_TARGETT17-
EXACT_MASS461.07152732799995Da
FORMULAC20H19N3O6S2-
HBA9-
HBD0-
LOGP2.778500000000001-
MOL_WEIGHT461.52100000000036g/mol
QED_SCORE0.5125594879910277-
ROTATABLE_BONDS6-
TPSA103.99000000000001A^2

Docking across targets

This compound is global in the current database. Below you can review all docking experiments and targets that contain imported poses for it, which is the basis for reverse docking analysis.

TargetExperimentReportPosesBest rankBest scoreNative overlapNative recallRMSD
T04 T04 selection_import_t04 1
native pose available
0.27097943228209714 -19.6635 13 0.68 - Best pose
T01 T01 selection_import_t01 1
native pose available
0.9544730494110983 -22.718 13 0.62 - Best pose
T17 T17 selection_import_t17 1
native pose available
1.2196504051403532 -21.3242 7 0.58 - Best pose
T02 T02 selection_import_t02 1
native pose available
1.3741049807450607 -20.44 14 0.67 - Best pose
T15 T15 selection_import_t15 1
native pose available
1.8007768117229013 -20.1444 11 0.85 - Best pose
T03 T03 selection_import_t03 2
native pose available
1.8058017168282356 -24.6674 13 0.65 - Best pose
T16 T16 selection_import_t16 2
native pose available
2.0182178879377184 -24.0955 5 0.42 - Best pose
T09 T09 selection_import_t09 1
native pose available
2.2832214801183897 -22.0808 13 0.62 - Best pose
T10 T10 selection_import_t10 3
native pose available
2.83121549954444 -22.7336 13 0.76 - Best pose
T12 T12 selection_import_t12 2
native pose available
2.8591163001678837 -22.5359 15 0.94 - Best pose
T13 T13 selection_import_t13 1
native pose available
3.435617077931159 -28.0542 14 0.74 - Best pose
T05 T05 selection_import_t05 1
native pose available
4.484716716621432 -28.8598 11 0.65 - Best pose
T04 — T04 1 poses · report selection_import_t04
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
458 0.27097943228209714 -0.811185 -19.6635 2 14 13 0.68 0.17 0.20 0.40 - no geometry warning; 8 clashes; 1 protein contact clash; 2 severe cofactor-context clashes Open pose
T01 — T01 1 poses · report selection_import_t01
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
513 0.9544730494110983 -0.848599 -22.718 5 16 13 0.62 0.00 0.00 0.00 - no geometry warning; 9 clashes; 4 protein contact clashes; 1 cofactor-context clash Open pose
T17 — T17 1 poses · report selection_import_t17
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
139 1.2196504051403532 -0.732121 -21.3242 5 16 7 0.58 0.00 0.00 0.00 - no geometry warning; 9 clashes; 5 protein contact clashes; moderate strain Δ 21.9 Open pose
T02 — T02 1 poses · report selection_import_t02
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
506 1.3741049807450607 -0.848148 -20.44 3 19 14 0.67 0.00 0.00 0.00 - no geometry warning; 9 clashes; 7 protein contact clashes; 1 cofactor-context clash Open pose
T15 — T15 1 poses · report selection_import_t15
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
114 1.8007768117229013 -0.767307 -20.1444 8 15 11 0.85 - - - - no geometry warning; 10 clashes; 9 protein contact clashes; moderate strain Δ 23.8 Open pose
T03 — T03 2 poses · report selection_import_t03
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
131 1.8058017168282356 -0.940039 -24.6674 6 14 13 0.65 0.29 0.20 0.20 - no geometry warning; 8 clashes; 1 protein clash; moderate strain Δ 23.5 Open pose
485 2.0994881049338083 -0.856427 -22.7639 4 13 9 0.45 0.29 0.20 0.20 - no geometry warning; 10 clashes; 1 protein clash Open pose
T16 — T16 2 poses · report selection_import_t16
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
117 2.0182178879377184 -0.829303 -24.0955 5 14 5 0.42 - - - - no geometry warning; 9 clashes; 1 protein clash; moderate strain Δ 23.6 Open pose
525 2.939096492500812 -0.773608 -21.4384 5 12 5 0.42 - - - - no geometry warning; 9 clashes; 2 protein clashes; moderate strain Δ 23.1 Open pose
T09 — T09 1 poses · report selection_import_t09
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
105 2.2832214801183897 -0.874039 -22.0808 4 17 13 0.62 0.00 0.00 0.00 - no geometry warning; 8 clashes; 1 protein clash; moderate strain Δ 21.1 Open pose
T10 — T10 3 poses · report selection_import_t10
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
453 2.83121549954444 -0.908661 -22.7336 12 15 13 0.76 0.62 0.55 0.64 - no geometry warning; 8 clashes; 1 protein clash; moderate strain Δ 20.9 Open pose
64 2.9866007130431282 -0.949521 -25.285 13 16 14 0.82 0.62 0.55 0.64 - no geometry warning; 9 clashes; 1 protein clash; moderate strain Δ 21.4 Open pose
91 3.5725886357035477 -0.950541 -26.1853 11 15 14 0.82 0.62 0.55 0.55 - no geometry warning; 8 clashes; 2 protein clashes; moderate strain Δ 23.7 Open pose
T12 — T12 2 poses · report selection_import_t12
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
447 2.8591163001678837 -0.882026 -22.5359 9 16 15 0.94 0.50 0.50 0.60 - no geometry warning; 8 clashes; 1 protein clash; moderate strain Δ 20.2 Open pose
89 3.588860201862459 -0.897555 -24.8412 10 10 8 0.50 0.42 0.30 0.30 - no geometry warning; 10 clashes; 2 protein clashes; moderate strain Δ 27.4 Open pose
T13 — T13 1 poses · report selection_import_t13
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
450 3.435617077931159 -1.00835 -28.0542 9 19 14 0.74 0.44 0.43 0.43 - no geometry warning; 9 clashes; 2 protein clashes Open pose
T05 — T05 1 poses · report selection_import_t05
Native comparison is calculated against the uploaded native ligand for the same experiment/target whenever it is available.
PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB strictHB roleHB residueRMSDExcludedNotes
425 4.484716716621432 -0.989791 -28.8598 6 13 11 0.65 0.14 0.17 0.40 - no geometry warning; 10 clashes; 3 protein clashes; 3 cofactor-context clashes Open pose
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Drug Similarity

Shared structural fragments with approved drugs — based on faircheckmol profile fingerprint.
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Structural Profile Fingerprint

Named-bit fingerprint from curated SMARTS patterns. Each bit = one chemical pattern.

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ADMET Profile

Computed from structure using RDKit. Indicative only — not a substitute for experimental data.

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3D Conformer

ETKDGv3 conformer generation with UFF minimisation. Rendered with 3Dmol.js.

This docking hit has a stored pose-level complex analysis page with clickable hydrogen bonds, π–π contacts, hydrophobic contacts, and clash inspection.
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